Custom Peptides
Cayman Chemical ArphamenIn BhemIsulfate 10mg
An aminopeptidase B inhibitor that is commonly used to characterize novel proteases
Cayman Chemical Schzndrn 10mg
A lignan with diverse biological activities; induces cell cycle arrest at the G0/G1 phase and inhibits growth of T47D and MDA-MB-231 breast cancer cells at 100 μM; prevents glutamate-induced cytotoxicity, inhibits production of NO and ROS, and preserves the mitochondrial membrane potential in isolated rat cortical cells at 10 and 100 μM; reduces cisplatin-induced apoptosis in HK-2 cells; reverses scopolamine-induced impairment of spatial memory and the passive avoidance response in rats at 1 and 10 mg/kg; enhances oxotremorine-induced tremors in mice; reduces serum levels of IgE, IgG1, IL-4, and IFN-γ in an ovalbumin-sensitized mouse model of allergy at 10 mg/kg
Cayman Chemical PerIndoprIlat 10mg
An ACE inhibitor (IC50 = 1.05 nM) and active metabolite of perindopril; reduces expression of the mRNA encoding VEGF in KB cells at 1 and 2 µM; induces endothelium-dependent relaxation in isolated dog basilar and coronary arteries (IC30s = 0.46 and 1.15 µM, respectively); reverses or prevents restricted oxygen-induced decreases in mean blood pressure, renal blood flow, and renal vascular resistance, as well as increases in the urine flow rate in an acute hypoxemia-induced rabbit model of renal hypoperfusion at 20 UG/kg
Cayman Chemical Isoxnthohumol 10mg
An enantiomer of isoxanthohumol; found in similar amounts as (+)-isoxanthohumol in beer
Cayman Chemical 4methoxyaPyrroldInopentIo 10mg
Shares structural features with the stimulant α-PVP, whose mechanism of action is unknown but is believed to act similarly to the designer drug MDPV
Cayman Chemical XE 991hydrochlorIde 10mg
A blocker of KCNQ channels that potently inhibits KCNQ1 and 2 homomeric channels (IC50 = 0.75 and 0.71 µM, respectively) as well as KCNQ2+3 heteromultimers (IC50 = 0.6 µM); shows good in vivo potency and duration of action
Cayman Chemical 1MyrIstyl2hydroxysnglyce 10mg
An LPA derivative and agonist of LPA1 and LPA2; increases calcium mobilization in a reporter assay using HEL 92.1.7 cells (EC50 = 37 nM)
Cayman Chemical 4-APBhydrochlorIde 10mg
An analytical reference standard categorized as a benzofuran; a potential metabolite of 4-MAPB and 4-EAPB based on the published metabolism of 5-MAPB; intended for research and forensic applications
Cayman Chemical DIltIazem-d3hydrochlorIde 10mg
An internal standard for the quantification of diltiazem by GC- or LC-MS
Cayman Chemical 15-keto Latnoprost 10mg
An active metabolite of latanoprost; intraocular administration reduces intraocular pressure in cynomolgus monkeys at 1 UG/eye; reduces pupillary diameter in cats when administered topically at 5 UG/eye
Cayman Chemical Solamargn 10mg
A glycoalkaloid with anticancer activity; decreases viability of H1650, H1975, PC-9, A549, and H1299 NSCLC cells at 6 µM; reduces tumor growth in an A549 mouse xenograft model at 8 mg/kg per day
Cayman Chemical 9 Z-Pentacosen 10mg
A cuticular hydrocarbon and insect sex hormone; found in the cuticle of female F. canicularis flies and is an attractant to males in a trap assay; a contact sex hormone in scarab beetles and locust borers that is more abundant in females than males; elicits arrestment, alignment, and mounting by males of both species in mating assays, but only elicits copulation by the locust borer; produced by the orchid O. exaltata and by C. cunicularius, a pollinator of O. exaltata